Mechano-activated GABA_B Receptor

GABA-independent

Mechanical forces directly activate GABA_B receptors without the neurotransmitter GABA, mediating astrocyte remodeling.

Huo, Yujia · Zhou, Yiwei · Lin, Li · Yang, Fan · Meng, Jiyong · He, Feiteng · Zhang, Fengfan · Shen, Cangsong · Liu, Yuxuan · Xu, Chanjuan · Xu, Shawn X.Z. · Liu, Jianfeng

Nature Communications 2025

Advantages

Shear stress promotes integrin binding to GB1

Induces allosteric rearrangement of GABA_B receptor transmembrane domains towards an active conformation

Shear stress-induced GABA_B receptor activation plays a crucial role in astrocyte remodeling